Publications

2022

Y. Hou, Y. Bando, D. Carrasco Flores, V. Hotter, B. Schiweck, T. Melzer, H.-D. Arndt, M. Mittag, "A cyclic lipopeptide produced by an antagonistic bacterium relies on its tail and TRP-type Ca2+ channels to immobilize a green alga", in revision

S. Lawrinowitz, J. M. Wurlitzer, D. Weiss, H.-D. Arndt, E. Kothe, M. Gressler, D. Hoffmeister, "Blue-Light-Dependent Pre-mRNA Splicing Controls Pigment Biosynthesis in the Mushroom Terana caerulea", Microbiol. Spectrum 2022, accepted

F. Küllmer, N. A. Vepřek, M. Borowiak, V. Nasufović, S. Barutzki, O. Thorn-Seshold, H.-D. Arndt, D. Trauner,"Next Generation Opto-Jasplakinolides Enable Local Remodeling of Actin Networks", Angew. Chem. 2022, accepted

Y. Bando, Y. Hou, L. Seyfarth, J. Probst, S. Gotze, M. Bogacz, U. A. Hellmich, P. Stallforth, M. Mittag, H. D. Arndt, "Total Synthesis and Structure Correction of the Cyclic Lipodepsipeptide Orfamide A"External link, Chem. Eur. J. 2022, 28, e202104417.

S. Dhiman, J. F. Ulrich, P. Wienecke, T. Wichard, H. D. Arndt, "Stereoselective Total Synthesis of (-)-Thallusin for Bioactivity ProfilingExternal link", Angew. Chem. Int. Ed. 2022, e202206746.

F. Kullmer, L. Gregor, H. D. Arndt, "Systematic modifications of substitution patterns for property tuning of photoswitchable asymmetric azobenzenesExternal link", Org. Biomol. Chem. 2022, 20, 4204-14.

A. Oberheide, F. Gaigne, H. D. Arndt, "Divergent Synthesis of C5-Heteroatom Substituted OxazolesExternal link", Adv. Synth. Catal. 2022, 364, 1903-7.

P. Wienecke, H. Goerls, H. D. Arndt, "Multigram-scale total synthesis of (-)-ambreinolide by a diastereoselective polyene cyclizationExternal link", Bioorg. Med. Chem. Lett. 2022, 72, 128845.

2021

S. Schwarthoff, N. Tischer, H. Sager, B. Schatz, M. M. Rohrbach, I. Raztsou, D. Robaa, F. Gaube, H. D. Arndt, T. Winckler, "Evaluation of gamma-carboline-phenothiazine conjugates as simultaneous NMDA receptor blockers and cholinesterase inhibitorsExternal link", Bioorg. Med. Chem. 2021, 46, 116355.

V. Nasufovic, F. Kullmer, J. Bossneck, H. M. Dahse, H. Gorls, P. Bellstedt, P. Stallforth, H. D. Arndt, "Total Synthesis and Bioactivity Mapping of Geodiamolide HExternal link", Chem. Eur. J. 2021, 27, 11633-42.

E. M. Molloy, M. Dell, V. G. Hansch, K. L. Dunbar, R. Feldmann, A. Oberheide, L. Seyfarth, J. Kumpfmuller, T. Horch, H. D. Arndt, C. Hertweck, "Enzyme-Primed Native Chemical Ligation Produces Autoinducing Cyclopeptides in ClostridiaExternal link", Angew. Chem. Int. Ed. 2021, 60, 10670-9.

S. Pospich, F. Küllmer, V. Nasufovic, J. Funk, A. Belvy, P. Bieling, H.-D. Arndt, S. Raunser, "Cryo-EM resolved molecular recognition of an optojasp photoswitch bound to actin filaments in both switch statesExternal link", Angew. Chem. 2021, 60, 8678-8682.

V. Nasufovic, P. Then, F. Dröge, M. Duong, B. Dietzek, R. Heintzmann, H.-D. Arndt, "Si-Rhodamine isothiocyanate as a fluorescent labeling toolExternal link", Org. Biomol. Chem. 2021, 19, 574-578.

2020

A. Oberheide, H.-D. Arndt, "Effective C5-arylation of peptide-integrated oxazoles: Almazole DExternal link", Adv. Synth. Catal. 2020, 363, 1132-1136.

R. R. A. Freund, M. van den Borg, D. Gassmaier, R. Schlosser, T. Jacob, H.-D. Arndt, "Cornforth-Evans transition states in stereocontrolled allylborations of epoxy aldehydesExternal link", Chem. Eur J. 2020, 26, 8639-8650.

M. Borowiak, F. Küllmer, F. Gegenfurtner, S. Peil, V. Nasufovic, S. Zahler, O. Thorn-Seshold, D. Trauner, H.-D. Arndt, "Optical manipulation of F-actin with photoswitchable small moleculesExternal link", J. Am. Chem. Soc. 2020, 142, 9240-9249 (press releaseExternal link of FSU Jena; featured on local radio SRBExternal link in GermanExternal link)

R. A. Freund, P. Gobrecht, D. Fischer, H.-D. Arndt, "Advances in parthenolide chemistry and biologyExternal link", Nat. Prod. Rep. 2020, 37, 541-565.

M. Sauer, V. Nasufovic, H.-D. Arndt, I. Vilotijevic, "Robust Synthesis of NIR-emissive P-Rhodamine FluorophoresExternal link", Org. Biomol. Chem. 2020, 18, 1567-1571.

 

2019

R. R. A. Freund, P. Gobrecht, P. Moser, D. Fischer, H.-D. Arndt, "Synthesis and biological profiling of parthenolide ether analogsExternal link", Org. Biomol. Chem. 2019, 17, 9703-9707.

A. Müller, S. Müller, V. Nasufovic, H.-D. Arndt, T. Pompe, "Actin stress fiber dynamics in laterally confined cellsExternal link", Integr. Biol. 2019, 11, 175-185.

R. R. A. Freund, P. Gobrecht, Z. Rao, J. Gerstmeier, R. Schlosser, H. Görls, O. Werz, D. Fischer, H.-D. Arndt, "Stereoselective total synthesis of parthenolides indicates target selectivity for tubulin carboxypeptidase activityExternal link", Chem. Sci. 2019, 10, 7358-7364.

A. Oberheide, S. Schwenk, C. Ronco, L.-M. Semmrau, H. Görls, H.-D. Arndt, "Synthesis, Structures, and Cytotoxicity of Urukthapelstatin A Polyazole Cyclopeptide AnalogsExternal link", Eur J. Org. Chem. 2019, 4320-4326 (cover featureExternal link: Eur J. Org. Chem. 2019, 4272).

S. Krieck, D. Kalden, A. Oberheide, L. Seyfarth, H.-D. Arndt, H. Görls, M. Westerhausen, "Synthesis and Catalytic Activity of Tridentate External linkN-(2-Pyridylethyl)-Substituted Bulky Amidinates of Calcium and StrontiumExternal link", Dalton Trans. 2019, 48, 2479-2490.

A. Oberheide, S. Pflanze, P. Stallforth, H.-D. Arndt, "Solid Phase Based Total Synthesis and Stereochemical Assignment of the Cryptic Natural Product AurantizolicinExternal link", Org. Lett. 2019, 21, 729-732.

2018

F. Merino, S. Pospich, J. Funk, F. Küllmer, H.-D. Arndt, P. Bieling, S. Raunser, "Structural transitions of F-actin upon ATP hydrolysis at near-atomic resolution revealed by cryo EMExternal link", Nat. Struct. Mol Biol. 2018, 25, 528-537.

C. Rößler, H.-D. Arndt, "A master switch in thiopeptide biosynthesisExternal link", Cell Chem. Biol. 2018, 25, 121-123.

 

2017

S. Zergiebel, H.-D. Arndt, A. Seeling, "Optimized Synthesis of new LE404-derived azecine-prodrugsExternal link", Tetrahedron Lett. 2017, 58, 3640-3642.

S. Zergiebel, C. Fleck, H.-D. Arndt, C. Enzensperger, A. Seeling, "Synthesis and Characterization of new Azecine-Derivatives as Potential NeurolepticsExternal link", Drug. Res. 2017, 67, 466-475.

K. B. Jadhav, C. Stein, O. Makarewicz, G. Pradel, R. J. Lichtenecker, H. Sack, S. H. Heinemann, H.-D. Arndt, "Bioactivity of topologically confined gramicidin A dimersExternal link", Bioorg. Med. Chem. 2017, 25, 261-268.

2016

Y. Yonemura, X. Li, K. Müller, A. Krämer, P. Atigbire, T. Mentrup, T. Feuerhake, T. Kroll, O. Shomron, R. Nohl, H.-D. Arndt, C. Hoischen, P. Hemmerich, K. Hirschberg, C. Kaether, "Inhibition of cargo export at ER-exit sites and the trans-Golgi network by the secretion inhibitor FLI-06External link", J. Cell. Sci. 2016, 129, 3868-3877.

R. R. A. Freund, H.-D. Arndt, "Synthesis of (±)-4,5-dia-parthenolide, an unnatural parthenolide stereoisomerExternal link", J. Org. Chem. 2016, 81, 11009-11016.

L. Gelis, N. Jovancevic, S. Veitinger, B. Mandal, H.-D. Arndt, E. M. Neuhaus, H. Hatt, "Functional characterization of the odorant receptor 51E2 in human melanocytesExternal link", J. Biol. Chem. 2016, 291, 17772-17786

K. P. Wojtas, J.-Y. Lu, D. Krahn, H.-D. Arndt, "Regioselective functionalization of 3-hydroxypyridine carboxylates by neighboring group assistanceExternal link", Chem. Asian J. 2016, 11, 2859-2862.

S. Schwenk, C. Ronco, A. Oberheide, H.-D. Arndt, "Biomimetic synthesis of urukthapelstatin A by Aza-Wittig ring contractionExternal link", Eur. J. Org. Chem. 2016, 4795-4799.

K. P. Wojtas, M. Riedrich, J.-Y. Lu, P. Winter, T. Winkler, S. Walter, H.-D. Arndt, "Total synthesis of nosiheptideExternal link", Angew. Chem. 2016, 128, 9924-9928; Angew. Chem. Int. Ed. 2016, 55, 9772-9776.

 

2015

H. B. Bode, A. O. Brachmann, K. B. Jadhav, L. Seyfarth, C. Dauth, S. W. Fuchs, M. Kaiser, N. R. Waterfield, H. Sack, S. H. Heinemann, H.-D. Arndt, "Structure elucidation and activity of the giant-NRPS derived D-/L-pentadecapeptide kolossin AExternal link", Angew. Chem. 2015, 127, 10493-10496; Angew. Chem. Int. Ed. 2015, 54, 10352-10355; Highlighted inExternal link Nachr. Chem. 2015, 63, 974.

K. B. Jadhav, R. J. Lichtenecker, A. Bullach, B. Mandal, H.-D. Arndt, "Dynamic combinatorial enrichment of polyconformational D-/L-peptide dimersExternal link", Chem. Eur. J. 2015, 21, 5898-5908.

H.-D. Arndt, S. Rizzo, C. Nöcker, V. N. Wakchaure, L.-G. Milroy, V. Bieker, A. Calderon, T. T. N. Tran, S. Brand, L. Dehmelt, H. Waldmann, "Covalent divergent solid-phase synthesis of natural product-inspired bipartite cyclodepsipeptides - Total synthesis of seragamide AExternal link", Chem. Eur. J. 2015, 21, 5311-5316.

 

2014

A. Wolf, S. Schoof, S. Baumann, H.-D. Arndt, K. N. Kirschner, "Structure-activity relationships of thiostrepton derivatives: Implications for rational drug designExternal link", J. Comput.-Aided Mol. Des. 2014, 28, 1205-1215.

G. Lukinavičius, L. Reymond, E. d'Este, A. Masharina, F. Göttfert, H. Ta, A. Güther, M. Fournier, S. Rizzo, H. Waldmann, C. Blaukopf, C. Sommer, D. W. Gerlich, H.-D. Arndt, S. W. Hell, K. Johnsson, "Fluorogenic probes for live-cell imaging of the cytoskeletonExternal link", Nat. Methods 2014, 11, 731-733.

2013

R. J. Lichtenecker, B. Ellinger, H.-M. Han, K. B. Jadhav, S. Baumann, O. Makarewicz, M. Grabenbauer, H.-D. Arndt, "Iterative antimicrobial candidate selection from informed D-/L-peptide librariesExternal link", ChemBioChem 2013, 14, 2492-2499.

A. Krämer, T. Mentrup, B. Kleizen, E. Rivera-Milla, D. Reichenbach, C. Enzensperger, R. Nohl, E. Täuscher, H. Görls, A. Ploubidou, C. Englert, O. Werz, H.-D. Arndt, C. Käther, "Small moleculesExternal link intercept Notch signalingExternal link and the early secretory pathwayExternal link", Nat. Chem. Biol. 2013, 9, 731-738.

J.-Y. Lu, M. Riedrich, K. P. Wojtas, H.-D. Arndt, "Assembly of the nosiheptide A-ring: A fruitful lessonExternal link", Synthesis 2013, 1300-1311.

P. Loos, C. Ronco, M. Riedrich, H.-D. Arndt, "Unified Azoline and Azole Syntheses by Optimized Aza-Wittig ChemistryExternal link", Eur. J. Org. Chem. 2013, 3290-3315.

 

2012

A. Wolf, S. Baumann, H.-D. Arndt, K. N. Kirschner, "Influence of thiostrepton binding on the ribosomal GTPase associated region characterized by molecular dynamics simulationExternal link", Bioorg. Med. Chem. 2012, 20, 7194-7205.

L.-G. Milroy, S. Rizzo, A. Calderon, B. Ellinger, S. Erdmann, J. Mondry, P. Verveer, P. Bastiaens, H. Waldmann, L. Dehmelt, H.-D. Arndt, "Selective chemical imaging of static actin in live cellsExternal link", J. Am. Chem. Soc. 2012, 134, 8480-8486.

M. N. Aminake, H.-D. Arndt, G. Pradel, "The proteasome of malaria parasites: a multi-stage drug target for chemotherapeutic intervention?External link", Int. J. Parasitol. Drugs Drug Res. 2012, 2, 1-10.

 

2011

L. Iovkova, D. Könning, B. Wängler, R. Schirrmacher, S. Schoof, H.-D. Arndt, K. Jurkschat, "SiFA-Modified Phenylalanine: A Key Compound for the Efficient Synthesis of External link¹⁸F-Labelled PeptidesExternal link", Eur. J. Inorg. Chem. 2011, 14, 2238-2246.

Y.-P. He, H. Tan, L. Arve, S. Baumann, H. Waldmann, H.-D. Arndt, "Biphenomycin B and Derivatives: Total Synthesis and Translation InhibitionExternal link", Chem. Asian J. 2011, 6, 1546-1556. 

S. Basu, B. Ellinger, S. Rizzo, C. Deraeve, M. Schürmann, H. Preut, H.-D. Arndt, H. Waldmann, "Biology-oriented synthesis of a natural-product inspired oxepane collection yields a small molecule activator of the Wnt-pathwayExternal link", Proc. Natl. Acad. Sci. USA 2011, 108, 6805-6810.

M. N. Aminake, S. Schoof, L. Sologub, M. Leubner, M. Kirschner, H.-D. Arndt, G. Pradel, "Thiostrepton and derivatives exhibit antimalarial and gametocytocidal activity by dually targeting the parasite proteasome and apicoplastExternal link", Antimicrob. Agents Chemother. 2011, 55, 1338-1348. 

H. R. A. Jonker, S. Baumann, A. Wolf, F. Hiller, S. Schoof, K. W. Schulte, K. N. Kirschner, H. Schwalbe, H.-D. Arndt, "NMR structures of thiostrepton derivatives reveal shape selective target recognitionExternal link", Angew. Chem. 2011, 123, 3366-3370; Angew. Chem. Int. Ed. 2011, 50, 3308-3312.

 

2010

S. Baumann, S. Schoof, M. Bolten, C. Haering, M. Takagi, K. Shin-ya, H.-D. Arndt, "Molecular determinants of microbial resistance to thiopeptide antibioticsExternal link", J. Am. Chem. Soc. 2010, 132, 6973-6981. 

C. P. R. Hackenberger, H.-D. Arndt, D. Schwarzer, "Semisynthese: Ein zentrales Werkzeug für die Chemische BiologieExternal link", Chem. Unserer Zeit 2010, 44, 198-206.

H.-D. Arndt, C. P. R. Hackenberger, D. Schwarzer, "Semisynthese: Chemie mit den Molekülen der NaturExternal link", Chem. Unserer Zeit 2010, 44, 130-137. 

S. Schoof, G. Pradel, M. N. Aminake, B. Ellinger, S. Baumann, M. Potowski, Y. Najajreh, M. Kirschner, H.-D. Arndt, "Anti-plasmodial thiostrepton derivatives are proteasome inhibitors with a dual mode of actionExternal link", Angew. Chem. 2010, 122, 3389-3393; Angew. Chem. Int. Ed. 2010, 49, 3317-3321. 

R. Tannert, L.-G. Milroy, T.-S. Hu, B. Ellinger, S. Menninger, H.-D. Arndt, H. Waldmann, "Synthesis and structure-activity correlation of natural-product inspired cytotoxic cyclodepsi­peptides stabilizing actinExternal link", J. Am. Chem. Soc. 2010, 132, 3063-3077.

 

2009

J.-Y. Lu, M. Riedrich, M. Mikyna, H.-D. Arndt, "Aza-Wittig-enabled synthesis of the nosiheptide A-RingExternal link", Angew. Chem. 2009, 121, 8281-8284; Angew. Chem. Int. Ed. 2009, 48, 8137-8140.

S. Schoof, H.-D. Arndt, "D-Cysteine occurrence in thiostrepton may not necessitate an epimeraseExternal link", Chem. Commun. 2009, 7113-7115.

H.-D. Arndt, S. Schoof, J.-Y. Lu, "Thiopeptide antibiotic biosynthesisExternal link", Angew. Chem. 2009, 121, 6900-6904; Angew. Chem. Int. Ed. 2009, 48, 6770-6773.

T. Walther, S. Renner, H. Waldmann, H.-D. Arndt, "Synthesis and structure-activity correlation of a brunsvicamide-inspired compound collectionExternal link", ChemBioChem 2009, 10, 1153-1162.

P. Loos, M. Riedrich, H.-D. Arndt, "AzaExternal link-Wittig access to chiral imidazol(in)esExternal link", Chem. Commun. 2009, 1900-1902 ("Highlight" in: Synfacts 2009, 7, 728).

R. Tannert, T.-S. Hu, H.-D. Arndt, H. Waldmann, "Solid-phase based total synthesis of jasplakinolide by ring-closing metathesisExternal link", Chem. Commun. 2009, 1493-1495.

B. Kilitoglu, H.-D. Arndt, "Scope of Tyrosine O-Arylations with Boronic Acids: Optimized Synthesis of an Orthogonally Protected IsodityrosineExternal link", Synlett 2009, 720-723.

S. Schoof, S. Baumann, B. Ellinger, H.-D. Arndt, "A fluorescent probe for the 70S-ribosomal GTPase-associated centerExternal link", ChemBioChem 2009, 10, 242-245.

 

2008

H. Waldmann, Y.-P. He, H. Tan, L. Arve, H.-D. Arndt, "Total synthesis of biphenomycin BExternal link", Chem. Commun. 2008, 5562-5564. 

J.-Y. Lu, J. Keith, W.-Z. Shen, M. Schürmann, H. Preut, T. Jacob, H.-D. Arndt, "Regioselective External linkde-novo synthesis of cyanohydroxy­pyridines with a concerted mechanismExternal link", J. Am. Chem. Soc. 2008, 130, 13219-13221. 

N. Bisek, S. Wetzel, H.-D. Arndt, H. Waldmann, "Synthesis and conformational analysis of stevastelin C3 analogs and their activity against the dual-specific phosphatase VHRExternal link", Chem. Eur. J. 2008, 14, 8847-8860.

H. Waldmann, T.-S. Hu, S. Renner, S. Menninger, R. Tannert, T. Oda, H.-D. Arndt, "Total synthesis of chondramide C and its binding mode to F-actinExternal link", Angew. Chem. 2008, 120, 6573-6577; Angew. Chem. Int. Ed. 2008, 47, 6473-6477.

S. Baumann, S. Schoof, S. D. Harkal, H.-D. Arndt, "Mapping the binding site of thiopeptide antibiotics by proximity induced covalent capture (PICC)External link", J. Am. Chem. Soc. 2008, 130, 5664-5666.

T. Walther, H.-D. Arndt, H. Waldmann, "Solid-support based total synthesis and stereochemical correction of brunsvicamide AExternal link", Org. Lett. 2008, 10, 3199-3202. 

H.-D. Arndt, M. Riedrich, "Synthesis of marine alkaloids from the oroidin familyExternal link", Angew. Chem. 2008, 120, 4864-4867; Angew. Chem. Int. Ed. 2008, 47, 4785-4788.

J.-Y. Lu, W.-Z. Shen, H. Preut, H.-D. Arndt, "(External linkZ)-Methyl-2-(methoxyimino)-3-oxo-butyrateExternal link", Acta. Cryst. E 2008, 64, o602.

 

2007

T.-S. Hu, R. Tannert, H.-D. Arndt, H. Waldmann, "Solid-phase based synthesis of jaspla­kinolide analogs by intramolecular azide/alkyne cycloadditionsExternal link", Chem. Commun. 2007, 3942-3944.

R. Tannert, M. Schürmann, H. Preut, H.-D. Arndt, H. Waldmann, "(External linkS)-3-((External linkR)-2,4-dimethylpent-4-enoyl)-4-isopropyl-5,5-diphenyloxazolidin-2-oneExternal link", Acta. Cryst. E 2007, 63, o4381.

H.-D. Arndt, S. Schoof, "Polyamide- and RNA-based activators in living cells: A major step towards controlling gene expressionExternal link", ChemBioChem 2007, 8, 1095-1098.

J.-Y. Lu, H.-D. Arndt, "Hetero-Diels-Alder synthesis of 3-hydroxypyridines: Access to the nosiheptide coreExternal link", J. Org. Chem. 2007, 72, 4205-4212.

M. Riedrich, S. D. Harkal, H.-D. Arndt, "Peptide-embedded heterocycles by mild single- and multiple External linkaza-Wittig ring closuresExternal link", Angew. Chem. 2007, 119, 2755-2758; Angew. Chem. Int. Ed. 2007, 46, 2701-2703.

R. L. Stafford, H.-D. Arndt, M. Brezinski, A. Ansari, P. B. Dervan, "Minimization of a DNA-protein dimerizerExternal link", J. Am. Chem. Soc. 2007, 129, 2660-2668. 

R. Wesolowski, A. Sommer, H.-D. Arndt, U. Koert, P. Reiß, S. Wimmers, O. Strauss, "Functional studies on synthetic gramicidin-hybrid ion channels in cellsExternal link", ChemBioChem 2007, 8, 513-520.

 

2006

H.-D. Arndt, "Small molecule modulators of transcriptionExternal link", Angew. Chem. 2006, 118, 4664-4673; Angew. Chem. Int. Ed. 2006, 45, 4552-4560.

 

Before 2006

K. E. Hauschild, R. E. Metzler, H.-D. Arndt, R. Moretti, M. Raffaelle, P. B. Dervan, A. Z. Ansari, "Temperature-sensitive protein-DNA dimerizersExternal link", Proc. Natl. Acad. Sci. USA 2005, 102, 5008-5013. 

Y. Kwon, H.-D. Arndt, Q. Mao, Y. Choi, Y. Kawazoe, P. B. Dervan, M. Uesugi, "A small molecule transcription factor mimicExternal link", J. Am. Chem. Soc. 2004, 126, 15940-15941.

H.-D. Arndt, B. Ziemer, U. Koert, "On the folding propensity of cyclohexylether-External linkδExternal link-peptidesExternal link", Org. Lett. 2004, 6, 3269-3271. 

H.-D. Arndt, R. Welz, S. Müller, B. Ziemer, U. Koert, "Stereoselective synthesis of External linktrans-External linkthreo-External linktrans oligo-pyrrolidines: Potential RNA cleavage agentsExternal link", Chem. Eur. J. 2004, 10, 3945-3962.

H.-D. Arndt, K. E. Hauschild, D. P. Sullivan, K. Lake, P. B. Dervan, A. Z. Ansari, "Toward artificial developmental regulatorsExternal link", J. Am. Chem. Soc. 2003, 125, 13322-13323.

H.-D. Arndt, D. Bockelmann, A. Knoll, S. Lamberth, C. Griesinger, U. Koert, "Cation control in functional helical programming: NMR-structures of a d-l-peptide ion channelExternal link", Angew. Chem. 2002, 114, 4234-4238; Angew. Chem. Int. Ed. 2002, 41, 4062-4065.

H.-D. Arndt, A. Vescovi, A. Schrey, J. R. Pfeifer, U. Koert, "Solution phase synthesis and purification of the minigramicidin ion channels and a succinyl-linked gramicidinExternal link", Tetrahedron 2002, 58, 2789-2801. 

H.-D. Arndt, A. Knoll, U. Koert, "Cyclohexylether-External linkδExternal link-amino acids: New selec­tivity fil­ters in ion channelsExternal link", Angew. Chem. 2001, 113, 2137-2140; Angew. Chem. Int. Ed. 2001, 40, 2076-2078.

H.-D. Arndt, A. Knoll, U. Koert, "Synthesis of minigramicidin ion channels and test of their hydrophobic match with the membraneExternal link", ChemBioChem 2001, 2, 221-223.

H.-D. Arndt, K. Polborn, U. Koert, "Stereoselective synthesis of a terpyrrolidine unit, a poten­tial building block for anion recognitionExternal link", Tetrahedron Lett. 1997, 38, 3879-3882.